SCHEMBL20052590

SCHEMBL20052590

O=C(CCl)NCCc1ccc(I)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.47
ST14 Q9Y5Y6 1/20 0.47
HPGD P15428 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
KDM4E B2RXH2 1/20 0.44
F13A1 P00488 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
CNR1 P21554 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28530111 0.85 ST14 (0.47) LMNAST14HPGDCA1CA2
SCHEMBL166076 0.84 ACACB (0.56) ST14HPGDKDM4EF13A1
SCHEMBL5574769 0.83 LMNA (0.66) LMNAHPGDCA1CA2TSHR
SCHEMBL2191045 0.83 KDM4E (0.65) LMNAKDM4EF13A1CYP1A2CYP2D6
SCHEMBL31248359 0.83 CA12 (0.49) LMNAHPGDCA1CA2CYP2C19
SCHEMBL9925290 0.81 HPGD (0.62) LMNAHPGDCNR1
SCHEMBL3316967 0.81 HPGD (0.68) LMNAHPGDCA1CA2TSHR
SCHEMBL6850677 0.81 ESRRG (0.53) LMNAST14HPGDCA1CA2
SCHEMBL2792326 0.81 HPGD (0.54) LMNAST14HPGDKDM4EF13A1
SCHEMBL696928 0.81 HDAC3 (0.62) HPGDCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944635-B2 Deuterated pyrazino[2,1-a]isoquinoline compounds and methods of treatment using the same CONCERT PHARMACEUTICALS, INC. (US) 2018-04-17 US disclosed