SCHEMBL20053619

SCHEMBL20053619

CC(C)(F)CN1CCC(COc2ccc(-c3ccc(C(=O)N4CCCC4)cc3)nc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.60
HRH3 Q9Y5N1 5/20 0.48
CYP4F2 P78329 6/20 0.44
CYP4A11 Q02928 6/20 0.44
RBP4 P02753 1/20 0.43
HPGDS O60760 1/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21534646 0.99 GPR119 (0.59) GPR119HRH3CYP4F2CYP4A11RBP4
SCHEMBL20053595 0.94 GPR119 (0.53) GPR119HRH3HPGDSHPGD
SCHEMBL15539154 0.92 GPR119 (0.53) GPR119HRH3CYP4F2CYP4A11HPGDS
SCHEMBL15538941 0.92 GPR119 (0.53) GPR119HRH3CYP4F2CYP4A11HPGDS
SCHEMBL15538942 0.92 GPR119 (0.53) GPR119HRH3CYP4F2CYP4A11HPGDS
SCHEMBL20053540 0.91 GPR119 (0.56) GPR119HRH3CYP4F2CYP4A11RBP4
SCHEMBL15537842 0.91 GPR119 (0.54) GPR119HRH3CYP4F2CYP4A11RBP4
SCHEMBL15539091 0.90 GPR119 (0.55) GPR119HRH3CYP4F2CYP4A11HPGDS
SCHEMBL15540121 0.90 GPR119 (0.55) GPR119HRH3CYP4F2CYP4A11HPGDS
SCHEMBL15539088 0.90 GPR119 (0.55) GPR119HRH3CYP4F2CYP4A11HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2858986-B1 PIPERIDINE DERIVATIVES AS GPR119 AGONISTS CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2019-10-30 EP disclosed
US-9944600-B2 Piperidine derivatives for GPR119 agonist CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2018-04-17 US disclosed