SCHEMBL20053810

SCHEMBL20053810

CSc1cn2ccccc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
RAB9A P51151 14/20 0.46
NPC1 O15118 13/20 0.46
KDM4E B2RXH2 6/20 0.45
PKM P14618 2/20 0.45
EPHX2 P34913 1/20 0.45
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 7/20 0.44
GFER P55789 2/20 0.44
ALOX12 P18054 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
MAPK1 P28482 2/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8185284 0.80 NPC1 (0.50) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL8189521 0.80 PTGS1 (0.44) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL6167210 0.79 PTGS1 (0.50) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL9517962 0.78 NPC1 (0.48) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL171008 0.74 PTGS1 (0.52) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL9517906 0.73 RAB9A (0.66) RAB9ANPC1KDM4EPKMSMN1; SMN2
SCHEMBL10333563 0.73 KDM4E (0.54) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL31731985 0.73 RAB9A (0.67) PTGS1PTGS2RAB9ANPC1KDM4E
SCHEMBL25150638 0.72 APP (0.32)
SCHEMBL22607307 0.72 HRH4 (0.42) KDM4EALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018237349-A1 INHIBITORS OF TYPED 1 METHIONYL-TRNA SYNTHETASE AND METHODS OF USING THEM UNIVERSITY OF WASHINGTON (US) 2018-12-27 WO claimed
US-9944644-B2 Octahydropyrrolopyrroles their preparation and use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-17 US disclosed