SCHEMBL20054511

SCHEMBL20054511

NCc1nc2ccc(C#Cc3ccc4nc(CN)[nH]c4c3)cc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.49
RAD52 P43351 1/20 0.47
UBE2N P61088 1/20 0.47
IDO1 P14902 1/20 0.47
KMT2A Q03164 4/20 0.47
POLB P06746 2/20 0.47
MAPT P10636 3/20 0.45
PKM P14618 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TPSAB1 Q15661 3/20 0.43
PRSS1 P07477 2/20 0.43
F2 P00734 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20054434 0.84 SCN10A (0.38) CACNA1HRAD52UBE2NIDO1KMT2A
Hydrochloric Acid SCHEMBL28836137 0.79 KMT2A (0.75) CACNA1HRAD52UBE2NIDO1KMT2A
SCHEMBL20054433 0.79 AAK1 (0.52) CACNA1HRAD52UBE2NIDO1KMT2A
SCHEMBL29409142 0.77 TDP1 (0.70) CACNA1HRAD52UBE2NIDO1KMT2A
SCHEMBL19377986 0.77 HDAC3 (0.52) CACNA1HRAD52UBE2NIDO1KMT2A
SCHEMBL4354084 0.77 TDP1 (0.70) CACNA1HRAD52UBE2NIDO1KMT2A
SCHEMBL38661663 0.77 IDO1 (0.76) CACNA1HRAD52UBE2NIDO1KMT2A
Hydrochloric Acid SCHEMBL23705615 0.76 HDAC3 (0.51) CACNA1HRAD52UBE2NIDO1KMT2A
Hydrochloric Acid SCHEMBL5204720 0.76 TDP1 (0.68) CACNA1HRAD52UBE2NIDO1KMT2A
Hydrochloric Acid SCHEMBL31164757 0.76 TDP1 (0.68) CACNA1HRAD52UBE2NIDO1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed