SCHEMBL20054531

SCHEMBL20054531

CC(C)(C)OC(=O)NC(c1ncc(C#Cc2ccc3cc(C#Cc4cnc(C(NC(=O)OC(C)(C)C)C(C)(C)C)[nH]4)ccc3c2)[nH]1)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.39
GABRG2 P18507 5/20 0.39
GABRB3 P28472 5/20 0.39
GABRA3 P34903 5/20 0.39
GABRA2 P47869 5/20 0.39
GABRB1 P18505 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA5 P31644 3/20 0.36
GABRA6 Q16445 3/20 0.36
GABRA4 P48169 2/20 0.36
TRPA1 O75762 2/20 0.35
PTPN1 P18031 2/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
SSTR3 P32745 1/20 0.34
AAK1 Q2M2I8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15116618 1.00 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL15125236 0.95 GABRA1 (0.36) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL16391245 0.94 GABRA1 (0.36) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL15116773 0.93 SSTR3 (0.39) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL20054356 0.93 SSTR3 (0.39) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL15116828 0.92 TRPA1 (0.38) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL16409154 0.87 SSTR3 (0.41) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL15125257 0.87 TRPA1 (0.35) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL15116615 0.84 TRPA1 (0.38) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL20054462 0.83 SSTR3 (0.40) GABRA1GABRG2GABRB3GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed