SCHEMBL20054612

SCHEMBL20054612

CCCN(C)CC(=O)Nc1ccc(C#Cc2ccc(NC)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
HPGD P15428 2/20 0.55
RAB9A P51151 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 2/20 0.51
NPC1 O15118 1/20 0.51
KMT2A Q03164 3/20 0.45
POLB P06746 1/20 0.45
MEN1 O00255 2/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP2C19 P33261 1/20 0.44
APP P05067 1/20 0.44
LTA4H P09960 4/20 0.43
GAA P10253 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
RORC P51449 2/20 0.42
ATM Q13315 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL400284 0.78 SMN1; SMN2 (0.65) ALDH1A1HPGDRAB9ASMN1; SMN2HTT
SCHEMBL13489789 0.78 KMT2A (0.49) ALDH1A1HPGDRAB9ASMN1; SMN2KMT2A
SCHEMBL20221643 0.78 RORC (0.52) ALDH1A1HPGDRAB9ASMN1; SMN2HTT
SCHEMBL403018 0.75 ALDH1A1 (0.41) ALDH1A1HPGDRAB9ASMN1; SMN2HTT
SCHEMBL404902 0.75 PPARG (0.41) ALDH1A1HPGD
SCHEMBL28939771 0.73 RAB9A (0.66) ALDH1A1HPGDRAB9ASMN1; SMN2HTT
SCHEMBL10915926 0.72 ALDH1A1 (0.54) ALDH1A1HPGDKMT2AMEN1CYP2C19
Hydrochloric Acid SCHEMBL10946080 0.71 ALDH1A1 (0.53) ALDH1A1HPGDKMT2AMEN1CYP2C19
SCHEMBL23222125 0.70 MAPT (0.83) ALDH1A1RAB9ASMN1; SMN2HTTKMT2A
SCHEMBL19002441 0.69 KMT2A (0.64) ALDH1A1RAB9ASMN1; SMN2NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed