SCHEMBL20059924

SCHEMBL20059924

COCCN/C(C)=C1\C(=N)CCCC1=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
GAA P10253 3/20 0.35
HPGD P15428 5/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
ALOX15 P16050 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
GLA P06280 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20060199 0.83 ALDH1A1 (0.33) ALDH1A1GAAHPGDHTTSMN1; SMN2
SCHEMBL20059969 0.82 ALDH1A1 (0.33) ALDH1A1GAAHPGDHTTSMN1; SMN2
SCHEMBL20060170 0.81 CNR2 (0.34) ALDH1A1GAAHPGDHTTSMN1; SMN2
SCHEMBL20060159 0.80 MEN1 (0.30) ALDH1A1MEN1KMT2A
SCHEMBL20059945 0.77 DPP7 (0.35) ALDH1A1HPGDKDM4E
SCHEMBL20059913 0.74
SCHEMBL20059935 0.72 HPGD (0.30) HPGDHTTSMN1; SMN2
SCHEMBL20060005 0.70
SCHEMBL20060140 0.66
SCHEMBL20059919 0.65 MEN1 (0.35) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed