SCHEMBL20064080

SCHEMBL20064080

CNC1CN(c2ncccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 2/20 0.39
HRH4 Q9H3N8 8/20 0.39
MAPT P10636 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDCD1LG2 Q9BQ51 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28250290 0.85 HRH4 (0.51) HRH3HRH4
SCHEMBL20064017 0.80 HRH4 (0.44) HRH3HRH4
SCHEMBL725763 0.80 KDM4E (0.51) KDM4EALDH1A1LMNAHRH4MAPT
SCHEMBL23023324 0.79 LMNA (0.47) KDM4EALDH1A1LMNAHRH4MAPT
SCHEMBL20283137 0.79 CHRM4 (0.41) HRH3KDM4EHRH4
Hydrochloric Acid SCHEMBL8695078 0.79 KDM4E (0.50) KDM4EALDH1A1LMNAHRH4MAPT
SCHEMBL29969592 0.77 KDM4E (0.49) HRH3KDM4EALDH1A1HRH4MAPT
SCHEMBL13703141 0.76 ALDH1A1 (0.43) KDM4EALDH1A1LMNAMAPTCYP2C19
SCHEMBL20283121 0.74 CHRM4 (0.47) HRH4
SCHEMBL24964199 0.74 HRH4 (0.53) HRH3KDM4EALDH1A1LMNAHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed