SCHEMBL20064413

SCHEMBL20064413

C=CCc1cc(O[C@H]2C[C@H](C(=O)NC3CN(c4ccnc(C)n4)C3)C2)c2ncsc2c1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.34
ACKR3 P25106 1/20 0.33
MALT1 Q9UDY8 1/20 0.30
SCN9A Q15858 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20064449 0.88 MALT1 (0.35) GPBAR1ACKR3MALT1SCN9A
SCHEMBL21222650 0.86 SCN9A (0.37) GPBAR1ACKR3MALT1SCN9A
SCHEMBL21222647 0.86 SCN9A (0.37) GPBAR1ACKR3MALT1SCN9A
SCHEMBL21222010 0.84 SCN9A (0.36) GPBAR1ACKR3MALT1SCN9A
SCHEMBL21222012 0.84 SCN9A (0.36) GPBAR1ACKR3MALT1SCN9A
SCHEMBL20064396 0.76 NPC1 (0.33)
SCHEMBL20064896 0.76 HCRTR2 (0.32) GPBAR1ACKR3
SCHEMBL20064062 0.75 PPARA (0.31)
SCHEMBL21222312 0.74 ACKR3 (0.38) ACKR3MALT1SCN9A
SCHEMBL21221932 0.74 SCN9A (0.39) ACKR3MALT1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed