SCHEMBL20064896

SCHEMBL20064896

C=CCc1cc(O[C@H]2C[C@H](C(=O)NC3CCN(c4ncc(F)cn4)CC3)C2)c2ncsc2c1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.32
SCD O00767 3/20 0.31
HPGD P15428 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ACKR3 P25106 2/20 0.30
GPBAR1 Q8TDU6 1/20 0.30
KDM1A O60341 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
KCNH2 Q12809 1/20 0.30
GPR119 Q8TDV5 1/20 0.30
F10 P00742 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21222419 0.89 HPGD (0.35) HCRTR2SCDHPGDALDH1A1MAPT
SCHEMBL21222416 0.89 HPGD (0.35) HCRTR2SCDHPGDALDH1A1MAPT
SCHEMBL21222128 0.82 ALDH1A1 (0.39) SCDHPGDALDH1A1MAPTSMN1; SMN2
SCHEMBL21222130 0.82 ALDH1A1 (0.39) SCDHPGDALDH1A1MAPTSMN1; SMN2
SCHEMBL21222019 0.81 CHRM4 (0.34) SCDHPGDALDH1A1MAPTSMN1; SMN2
SCHEMBL21222017 0.81 CHRM4 (0.34) SCDHPGDALDH1A1MAPTSMN1; SMN2
SCHEMBL21222336 0.79 HDAC3 (0.32) ACKR3HDAC6
SCHEMBL21222339 0.79 HDAC3 (0.32) ACKR3HDAC6
SCHEMBL20064062 0.76 PPARA (0.31)
SCHEMBL20064413 0.76 GPBAR1 (0.34) ACKR3GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed