SCHEMBL20064449

SCHEMBL20064449

Cc1cc(OC2CC(C(=O)NC3CN(c4ccnc(C)n4)C3)C2)c2ncsc2c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
ACKR3 P25106 1/20 0.34
SCN9A Q15858 7/20 0.33
RAB9A P51151 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HSD17B10 Q99714 2/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21222647 0.93 SCN9A (0.37) MALT1GPBAR1ACKR3SCN9AHCRTR1
SCHEMBL21222650 0.93 SCN9A (0.37) MALT1GPBAR1ACKR3SCN9AHCRTR1
SCHEMBL21222010 0.90 SCN9A (0.36) MALT1GPBAR1ACKR3SCN9AHCRTR1
SCHEMBL21222012 0.90 SCN9A (0.36) MALT1GPBAR1ACKR3SCN9AHCRTR1
SCHEMBL20064413 0.88 GPBAR1 (0.34) MALT1GPBAR1ACKR3SCN9A
SCHEMBL20064528 0.80 SCN9A (0.37) MALT1SCN9A
SCHEMBL21222312 0.80 ACKR3 (0.38) MALT1ACKR3SCN9ACCNCCDK8
SCHEMBL21221932 0.80 SCN9A (0.39) MALT1ACKR3SCN9AHCRTR1HCRTR2
SCHEMBL21222321 0.80 SLC6A9 (0.33) MALT1ACKR3
SCHEMBL21222322 0.80 SLC6A9 (0.33) MALT1ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed