SCHEMBL2007371

SCHEMBL2007371

COc1ccc2c(c1)c(C(=O)c1ccc(-c3cccnc3)s1)cn2Cc1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.48
ALDH1A1 P00352 2/20 0.47
AHR P35869 1/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.43
SERPINE1 P05121 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
ROCK2 O75116 1/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
PLA2G2A P14555 2/20 0.41
PTGS2 P35354 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYP17A1 P05093 1/20 0.41
CYP11B1 P15538 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005436 0.91 LMNA (0.48) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2012914 0.91 LMNA (0.56) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2002885 0.90 LMNA (0.47) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2002890 0.88 AHR (0.49) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2002871 0.86 LMNA (0.53) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL1999240 0.85 IRAK4 (0.51) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2002672 0.85 LMNA (0.48) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2006000 0.85 LMNA (0.48) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2000164 0.84 AHR (0.50) LMNAALDH1A1AHRMAPTSMN1; SMN2
SCHEMBL2007180 0.83 PLA2G2A (0.50) LMNAALDH1A1MAPTHSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed