SCHEMBL2002890

SCHEMBL2002890

COc1ccc2c(c1)c(C(=O)c1nnc(-c3cccnc3)s1)cn2Cc1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.49
LMNA P02545 3/20 0.47
ALDH1A1 P00352 3/20 0.46
MAPT P10636 2/20 0.44
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
SERPINE1 P05121 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
KDM4E B2RXH2 1/20 0.42
PTGS2 P35354 2/20 0.41
PLA2G2A P14555 1/20 0.41
CYP17A1 P05093 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012463 0.92 LMNA (0.56) AHRLMNAALDH1A1MAPTKMT2A
SCHEMBL2004829 0.91 AHR (0.50) AHRLMNAALDH1A1MAPTKMT2A
SCHEMBL2002885 0.88 LMNA (0.47) AHRLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL2007371 0.88 LMNA (0.48) AHRLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL2004404 0.87 AHR (0.49) AHRLMNAALDH1A1MAPTKMT2A
SCHEMBL1999240 0.86 IRAK4 (0.51) AHRLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL2000164 0.86 AHR (0.50) AHRLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL1998380 0.86 AHR (0.49) AHRLMNAALDH1A1MAPTKMT2A
SCHEMBL2004951 0.84 AHR (0.54) AHRLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL2003656 0.84 AHR (0.49) AHRLMNAALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed