SCHEMBL20076233

SCHEMBL20076233

COC(=O)c1c(F)cc(CCNCCNC(=O)OC(C)(C)C)cc1F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.39
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
NAMPT P43490 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
MALT1 Q9UDY8 1/20 0.36
IDO1 P14902 1/20 0.36
DRD2 P14416 1/20 0.35
GAA P10253 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGER4 P35408 1/20 0.35
POLB P06746 1/20 0.35
EPHX1 P07099 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399537 0.82 CA1 (0.43) NQO2CA1CA2NAMPTMALT1
SCHEMBL30754099 0.82 APLNR (0.36) NQO2CA1CA2GAA
SCHEMBL5109167 0.81 CA1 (0.43) NQO2CA1CA2TDP1NAMPT
SCHEMBL5109992 0.80 CA2 (0.45) NQO2CA1CA2TDP1NAMPT
SCHEMBL19300685 0.79 TACR1 (0.44) NQO2CA1CA2TDP1NAMPT
SCHEMBL3696922 0.78 NQO2 (0.47) NQO2CA1CA2TDP1NAMPT
SCHEMBL8401477 0.77 CTSS (0.50) NQO2NAMPTIDO1MEN1KMT2A
SCHEMBL23684682 0.75 CACNA1H (0.42) NQO2CA1CA2DRD2MEN1
SCHEMBL19026304 0.75 CA1 (0.41) NQO2CA1CA2TDP1NAMPT
SCHEMBL8399561 0.75 IDO1 (0.55) CA1CA2NAMPTMALT1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071606-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR Arvinas, Inc. (US) 2018-04-19 WO disclosed