SCHEMBL20095950

SCHEMBL20095950

C=CCCc1ccc(Br)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.41
LMNA P02545 2/20 0.41
PYCR1 P32322 1/20 0.41
HPGD P15428 3/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
SLC6A2 P23975 1/20 0.33
ADRA1D P25100 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17713325 0.81 PYCR1 (0.41) HTTLMNAPYCR1HPGDNPC1
SCHEMBL8173928 0.81 LMNA (0.43) HTTLMNAPYCR1HPGDNPC1
SCHEMBL248224 0.81 IDO1 (0.50) HTTHPGDTP53ALDH1A1IDO1
SCHEMBL30271268 0.81 IDO1 (0.50) HTTHPGDTP53ALDH1A1IDO1
SCHEMBL27519718 0.76 PYCR1 (0.45) HTTLMNAPYCR1NPC1RAB9A
SCHEMBL20801052 0.75 HPGD (0.38) HTTLMNAPYCR1HPGDNPC1
SCHEMBL1569794 0.75 TAAR1 (0.52) PYCR1HTR2AHRH1
SCHEMBL32689207 0.75 TAAR1 (0.52) PYCR1HTR2AHRH1
SCHEMBL11452260 0.75 PYCR1 (0.51) PYCR1HPGDHTR2ASLC6A4ALDH1A1
SCHEMBL589200 0.75 PYCR1 (0.44) HTTLMNAPYCR1SMN1; SMN2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018072602-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2018-04-26 WO disclosed