SCHEMBL20095956

SCHEMBL20095956

Cc1cc(F)c(Br)c(C#N)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.37
CYP11B2 P19099 4/20 0.37
TRPV4 Q9HBA0 2/20 0.36
MAOB P27338 2/20 0.34
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
MAOA P21397 1/20 0.34
AR P10275 3/20 0.33
DHODH Q02127 1/20 0.32
KHK P50053 1/20 0.32
TSHR P16473 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
EGLN2 Q96KS0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14033196 0.78 TRPV4 (0.39) CYP11B1CYP11B2TRPV4ESR1ESR2
SCHEMBL405549 0.78 TRPV4 (0.39) CYP11B1CYP11B2TRPV4ESR1ESR2
SCHEMBL2651893 0.78 TRPV4 (0.39) CYP11B1CYP11B2TRPV4MAOBESR1
SCHEMBL8062622 0.77 KDM1A (0.39) TSHRALDH1A1
SCHEMBL17185578 0.75 DHODH (0.35) CYP11B1CYP11B2TRPV4MAOBMAOA
SCHEMBL14744326 0.75 KHK (0.39) CYP11B1CYP11B2TRPV4ESR1ESR2
SCHEMBL404723 0.75 ADRB2 (0.45) CYP11B1CYP11B2TRPV4ARDHODH
SCHEMBL13855817 0.75 SELL (0.41) CYP11B1CYP11B2TRPV4ESR1ESR2
SCHEMBL22119927 0.75 KHK (0.39) CYP11B1CYP11B2TRPV4MAOBESR1
SCHEMBL29490392 0.75 DHODH (0.35) CYP11B1CYP11B2TRPV4MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018075871-A1 NOVEL ANTIBIOTICS AND METHODS OF USING SAME THE BROAD INSTITUTE, INC. (US) 2018-04-26 WO disclosed