SCHEMBL2009654

SCHEMBL2009654

COc1c(C(=O)OCc2ccccc2)cccc1S(=O)(=O)Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
TDP1 Q9NUW8 3/20 0.50
L3MBTL1 Q9Y468 4/20 0.48
TSHR P16473 2/20 0.48
CYP3A4 P08684 2/20 0.48
MAPK1 P28482 1/20 0.48
RAB9A P51151 2/20 0.47
CASP3 P42574 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
POLB P06746 2/20 0.47
KMT2A Q03164 2/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
MEN1 O00255 1/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3894645 0.85 ALDH1A1 (0.61) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL2007420 0.84 ALDH1A1 (0.54) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL12569669 0.83 ALDH1A1 (0.55) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL23183003 0.81 ALDH1A1 (0.59) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL28171736 0.80 RAB9A (0.65) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL2004907 0.79 F2 (0.47) ALDH1A1TDP1TSHRMAPK1KMT2A
Hydrochloric Acid SCHEMBL2008786 0.77 ALDH1A1 (0.55) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL20083681 0.76 ALDH1A1 (0.61) ALDH1A1TDP1L3MBTL1TSHRCYP3A4
SCHEMBL2005291 0.76 CA1 (0.39) ALDH1A1RAB9AKDM4ENPC1NPSR1
SCHEMBL14395398 0.75 ALDH1A1 (0.63) ALDH1A1TDP1L3MBTL1TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1864976-B1 PROPANE-1,3-DION DERIVATIVE OR SALT THEREOF ASTELLAS PHARMA INC (JP) 2012-10-10 EP disclosed
US-7960562-B2 Propane-1,3-dione derivative or salt thereof ASTELLAS PHARMA INC. (JP) 2011-06-14 US disclosed
CN-101142193-B 1, 3-propanedione derivative or salt thereof ASTELLAS PHARMA INC 2010-12-29 CN disclosed
US-20090181964-A1 Propane-1,3-Dione Derivative or Salt Thereof ASTELLAS PHARMA INC. 2009-07-16 US disclosed
CN-101142193-A 1, 3-propanedione derivative or salt thereof ASTELLAS PHARMA INC (JP) 2008-03-12 CN disclosed
EP-1864976-A1 PROPANE-1,3-DION DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2007-12-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090181964-A1 Propane-1,3-Dione Derivative or Salt Thereof GNRHR, KISS1R, FSHR ALDH1A1 2646/4885TDP1 3230/4885L3MBTL1 4375/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.