SCHEMBL20099962

SCHEMBL20099962

O[C@H](CF)CCn1cccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
FDPS P14324 1/20 0.40
DAO P14920 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
LMNA P02545 3/20 0.33
POLB P06746 1/20 0.33
THRB P10828 2/20 0.32
IDO1 P14902 1/20 0.31
HTT P42858 2/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
GAA P10253 2/20 0.30
ALDH1A1 P00352 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
KDM5A P29375 1/20 0.30
KDM2B Q8NHM5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20099935 0.83 TSHR (0.42) TSHRFDPSDAOADRB2ADRB1
SCHEMBL21996528 0.82 TSHR (0.44) TSHRFDPSDAOADRB2ADRB1
SCHEMBL31581978 0.82 TSHR (0.44) TSHRFDPSDAOADRB2ADRB1
SCHEMBL20099857 0.77 TSHR (0.38) TSHRFDPSDAOADRB2ADRB1
SCHEMBL20099882 0.74 LMNA (0.34) TSHRFDPSDAOL3MBTL1LMNA
SCHEMBL12181347 0.73
SCHEMBL27841918 0.73 TSHR (0.44) TSHRFDPSDAOLMNATHRB
SCHEMBL278529 0.72 L3MBTL1 (0.48) TSHRFDPSDAOL3MBTL1LMNA
SCHEMBL5713341 0.72 DAO (0.50) TSHRFDPSDAOLMNAPOLB
SCHEMBL3768453 0.71 TSHR (0.58) TSHRFDPSDAOADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3315492-A1 PYRAZOLE DERIVATIVE, OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Kissei Pharmaceutical Co., Ltd. (JP) 2018-05-02 EP disclosed