SCHEMBL20103203

SCHEMBL20103203

O=C(N[C@H]1CC[C@@]2(CCN(c3ccc(F)cc3Cl)C2=O)CC1)c1ccccn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.44
GAA P10253 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GRM4 Q14833 6/20 0.44
GRM5 P41594 4/20 0.43
PDE4B Q07343 1/20 0.42
GRM1 Q13255 2/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 1/20 0.41
TNKS2 Q9H2K2 2/20 0.41
TNKS O95271 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103129 0.88 SMYD3 (0.49) SMYD3GAAKMT2AGRM4GRM5
SCHEMBL20103437 0.86 HTR2A (0.39) GAAKMT2ASMN1; SMN2PDE4BHPGD
SCHEMBL20103204 0.84 PDE4B (0.44) PDE4BHPGDTNKS2TNKS
SCHEMBL18216338 0.83 HPGD (0.46) SMN1; SMN2PDE4BHPGDALDH1A1
SCHEMBL20103078 0.83 HPGD (0.54) KMT2ASMN1; SMN2GRM4PDE4BHPGD
SCHEMBL20103438 0.83 LMNA (0.44) KMT2APDE4BHPGDTNKS2TNKS
SCHEMBL18208311 0.82 KMT2A (0.42) KMT2APDE4BHPGDALDH1A1
SCHEMBL18208313 0.82 KMT2A (0.42) KMT2APDE4BHPGDALDH1A1
SCHEMBL18209065 0.82 IRAK4 (0.49) KDM4ETNKSHSD17B10
SCHEMBL18208502 0.82 IRAK4 (0.49) KDM4ETNKSHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078005-A1 AMIDO-SUBSTITUTED AZASPIRO DERIVATIVES AS TANKYRASE INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed