SCHEMBL20103692

SCHEMBL20103692

Cc1ccc(CNCCc2cccc3cc[nH]c23)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.52
HTR2C P28335 1/20 0.52
CHRM2 P08172 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
MPO P05164 2/20 0.39
MC5R P33032 1/20 0.39
MC3R P41968 1/20 0.39
MC1R Q01726 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38
AR P10275 1/20 0.38
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17118054 0.86 HTR2A (0.49) HTR2AHTR2CCHRM2CA12CA1
SCHEMBL16806760 0.77 HDAC1 (0.60)
SCHEMBL16806754 0.77 HTR2A (0.44) HTR2AHTR2CKMT2A
SCHEMBL2263387 0.76 HTR2A (0.48) HTR2AHTR2CMPONR3C1PGR
SCHEMBL5948742 0.74 NR3C1 (0.48) NR3C1PGRNR3C2ARMEN1
SCHEMBL2260650 0.74 HTR2A (0.55) HTR2AHTR2CNR3C1PGRNR3C2
SCHEMBL4985160 0.74 PKM (0.47) HTR2AHTR2CMC5RMC1RMEN1
SCHEMBL2260646 0.73 HTR2A (0.46) HTR2AHTR2CNR3C1PGRNR3C2
SCHEMBL31369960 0.72 KEAP1 (0.46) HTR2AHTR2CNR3C1PGRNR3C2
SCHEMBL16806761 0.72 HDAC1 (0.41) HTR2AHTR2CMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3110810-B1 PYRAZOLE AMIDE DERIVATIVE TEIJIN PHARMA LTD (JP) 2018-05-02 EP disclosed