SCHEMBL20103822

SCHEMBL20103822

O=C(Nc1ccc(CCc2nc3ccccc3[nH]2)cc1)Nc1cccc(C(F)(F)F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 18/20 1.00
NTRK2 Q16620 14/20 1.00
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
MTOR P42345 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103543 0.86 NTRK1 (0.84) NTRK1NTRK2NPC1RAB9A
SCHEMBL20103636 0.85 NTRK1 (1.00) NTRK1NTRK2NPC1RAB9A
SCHEMBL20103744 0.83 NTRK1 (0.79) NTRK1NTRK2
SCHEMBL20103646 0.82 NTRK1 (1.00) NTRK1NTRK2NPC1RAB9A
SCHEMBL30933634 0.81 MTOR (0.76) NTRK1NTRK2NPC1RAB9AMTOR
SCHEMBL20103766 0.81 NTRK1 (0.82) NTRK1NTRK2NPC1RAB9A
SCHEMBL7136568 0.79 NTRK1 (0.66) NTRK1NTRK2NPC1RAB9A
SCHEMBL21581198 0.79 NTRK1 (0.66) NTRK1NTRK2NPC1RAB9A
SCHEMBL20103644 0.78 NTRK1 (0.83) NTRK1NTRK2NPC1RAB9A
SCHEMBL6801623 0.77 NTRK1 (0.62) NTRK1NTRK2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed