SCHEMBL20103644

SCHEMBL20103644

COc1ccc(NC(=O)Nc2ccc(CCc3nc4ccccc4[nH]3)cc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 17/20 0.83
NTRK2 Q16620 13/20 0.80
MEN1 O00255 1/20 0.69
ALDH1A1 P00352 1/20 0.69
POLB P06746 1/20 0.69
KMT2A Q03164 1/20 0.69
TDP1 Q9NUW8 1/20 0.69
THRB P10828 1/20 0.60
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103646 0.91 NTRK1 (1.00) NTRK1NTRK2MEN1KMT2ANPC1
SCHEMBL20103543 0.88 NTRK1 (0.84) NTRK1NTRK2NPC1RAB9A
SCHEMBL20103744 0.85 NTRK1 (0.79) NTRK1NTRK2ALDH1A1
SCHEMBL20103766 0.85 NTRK1 (0.82) NTRK1NTRK2NPC1RAB9A
SCHEMBL27093086 0.81 RAB9A (0.71) MEN1ALDH1A1POLBKMT2ATDP1
SCHEMBL30933630 0.81 RAB9A (0.71) MEN1ALDH1A1POLBKMT2ATDP1
SCHEMBL20103636 0.81 NTRK1 (1.00) NTRK1NTRK2NPC1RAB9A
SCHEMBL25334690 0.80 NPC1 (0.64) NTRK1MEN1ALDH1A1POLBKMT2A
SCHEMBL32680055 0.80 NPC1 (0.64) NTRK1MEN1ALDH1A1POLBKMT2A
SCHEMBL20103822 0.78 NTRK1 (1.00) NTRK1NTRK2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed