SCHEMBL2010387

SCHEMBL2010387

Cc1[nH]c(=O)c(-c2ccccc2)c(C(F)(F)F)c1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.45
GRM6 O15303 1/20 0.43
ALDH1A1 P00352 5/20 0.41
RAB9A P51151 2/20 0.41
HTT P42858 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRA6 Q16445 1/20 0.35
MDM2 Q00987 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30472331 0.73 NR4A2 (0.48) LMNAGRM6ALDH1A1RAB9AHTT
SCHEMBL29031850 0.73 NR4A2 (0.48) LMNAGRM6ALDH1A1RAB9AHTT
SCHEMBL28768946 0.70 IGF1R (0.39) ALDH1A1NPSR1POLBMAPTHPGD
SCHEMBL2012056 0.68 LMNA (0.50) LMNAALDH1A1RAB9ASMN1; SMN2PDE4A
SCHEMBL15579812 0.68 AR (0.36) GRM6NPSR1GABRA1GABRG2GABRB3
SCHEMBL2431068 0.68 AR (0.36) GRM6ALDH1A1GABRA1GABRG2GABRB3
SCHEMBL28046061 0.67 FABP4 (0.35) LMNAGRM6ALDH1A1RAB9ANPSR1
SCHEMBL12293219 0.67 AR (0.34) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL15174105 0.66 NR4A2 (0.69) LMNAALDH1A1RAB9AHTTNPSR1
SCHEMBL27987654 0.66 GRM6 (0.45) LMNAGRM6ALDH1A1RAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513061-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2012-10-24 EP disclosed
WO-2011072691-A1 PYRIDONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2011-06-23 WO disclosed