SCHEMBL2002120

SCHEMBL2002120

COc1ccc2c(c1)c(C(=O)c1nc(-c3cccnc3)no1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
LMNA P02545 2/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 4/20 0.38
TP53 P04637 4/20 0.38
GSK3B P49841 2/20 0.38
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
RET P07949 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
PKM P14618 2/20 0.37
CYP3A4 P08684 2/20 0.37
PLA2G2A P14555 2/20 0.37
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002951 0.94 S1PR1 (0.41) ABCB1ABCC1ABCG2LMNATSHR
SCHEMBL2005430 0.94 LMNA (0.41) LMNATSHRMAPK1L3MBTL1MAPT
SCHEMBL2005843 0.91 GSK3B (0.40) LMNATSHRMAPK1L3MBTL1MAPT
SCHEMBL2007930 0.91 PLA2G2A (0.38) LMNATSHRL3MBTL1MAPTTP53
SCHEMBL2004518 0.91 ABCB1 (0.42) ABCB1ABCC1ABCG2LMNATSHR
SCHEMBL2000312 0.91 LMNA (0.39) LMNATSHRMAPK1L3MBTL1MAPT
SCHEMBL2001925 0.91 LMNA (0.41) ABCB1ABCC1ABCG2LMNATSHR
SCHEMBL2008765 0.90 PLA2G2A (0.42) LMNATSHRMAPK1L3MBTL1MAPT
SCHEMBL2002228 0.90 LMNA (0.40) LMNATSHRMAPK1L3MBTL1MAPT
SCHEMBL2010388 0.89 MAPT (0.39) ABCB1ABCC1ABCG2LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed