SCHEMBL2010576

SCHEMBL2010576

Nc1cccc2c1CNC2C1CCC(=O)NC1=O

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 20/20 0.48
DDB1 Q16531 15/20 0.48
TNF P01375 3/20 0.48
IL1B P01584 3/20 0.48
IKZF3 Q9UKT9 3/20 0.48
IKZF1 Q13422 2/20 0.48
BRD4 O60885 1/20 0.48
TBXA2R P21731 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31292137 0.84 CRBN (0.46) CRBNDDB1TNFIL1BIKZF3
SCHEMBL1897413 0.80 CRBN (0.45) CRBNDDB1TNFIL1BIKZF3
SCHEMBL6180923 0.78 CRBN (0.46) CRBNDDB1IKZF3
SCHEMBL27479960 0.78 CRBN (0.46) CRBNDDB1IKZF3
SCHEMBL8058860 0.76 CRBN (0.48) CRBNDDB1IKZF3
SCHEMBL3965614 0.76 CRBN (0.47) CRBNDDB1TNFIL1BIKZF3
SCHEMBL10192652 0.73 CRBN (0.53) CRBNDDB1TNFIL1BIKZF3
SCHEMBL21843690 0.73 CRBN (0.49) CRBNDDB1TNFIL1BIKZF3
SCHEMBL10192664 0.73 CRBN (0.53) CRBNDDB1TNFIL1BIKZF3
SCHEMBL2148301 0.71 CRBN (0.47) CRBNDDB1TNFIL1BIKZF3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504703-A1 IMMUNOMODULATORY COMPOUNDS FOR THE RESTORATION OF VITAMIN D SENSITIVITY IN VITAMIN D RESISTANT TUMOR CELLS Celgene Corporation (US) 2012-10-03 EP disclosed
WO-2011066351-A1 IMMUNOMODULATORY COMPOUNDS FOR THE RESTORATION OF VITAMIN D SENSITIVITY IN VITAMIN D RESISTANT TUMOR CELLS CELGENE CORPORATION (US) 2011-06-03 WO disclosed
EP-2235535-A2 BIOMARKERS FOR PREDICTING THE SENSITIVITY OF CELLS TO IMMUNOMODULATORY COMPOUNDS DURING TREATMENT OF NON-HODGKIN'S LYMPHOMA CELGENE CORPORATION (US) 2010-10-06 EP disclosed
WO-2009105256-A2 METHOD OF TREATING CANCER BY ADMINISTERING AN IMMUNOMODULATORY COMPOUND IN COMBINATION WITH A CD40 ANTIBODY OR CD40 LIGAND CELGENE CORPORATION (US) 2009-08-27 WO disclosed
WO-2009075797-A2 BIOMARKERS FOR PREDICTING THE SENSITIVITY OF CELLS TO IMMUNOMODULATORY COMPOUNDS DURING TREATMENT OF NON-HODGKIN'S LYMPHOMA CELGENE CORPORATION (US) 2009-06-18 WO disclosed