SCHEMBL2010739

SCHEMBL2010739

CCOc1c(C#N)ccc(-c2ccccc2)c1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 1/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 5/20 0.37
L3MBTL1 Q9Y468 3/20 0.37
HPGD P15428 3/20 0.37
ALDH1A1 P00352 8/20 0.36
TDP1 Q9NUW8 4/20 0.36
GAA P10253 2/20 0.36
POLB P06746 1/20 0.36
GALR3 O60755 1/20 0.35
SQOR Q9Y6N5 2/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
MAPT P10636 2/20 0.35
SCN9A Q15858 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8001576 0.80 GRIN2D (0.46) HPRT1LMNAKDM4EHPGDALDH1A1
SCHEMBL10337978 0.74 ALDH1A1 (0.49) HPRT1KDM4EHPGDALDH1A1TDP1
SCHEMBL30204899 0.73 LMNA (0.50) LMNAHPGDALDH1A1TDP1POLB
SCHEMBL9829866 0.73 LMNA (0.50) LMNAHPGDALDH1A1TDP1POLB
SCHEMBL8197182 0.72 PTGDR2 (0.41) HPRT1LMNAKDM4EL3MBTL1HPGD
SCHEMBL29192937 0.72 HTT (0.42) HPRT1LMNAKDM4EHPGDALDH1A1
SCHEMBL29193181 0.71 XDH (0.40) HPRT1KDM4EHPGDALDH1A1TDP1
SCHEMBL3577756 0.71 AR (0.43)
SCHEMBL29236231 0.71 ALDH1A1 (0.59) HPRT1LMNAALDH1A1TDP1POLB
SCHEMBL11292185 0.71 ALDH1A1 (0.57) LMNAKDM4EALDH1A1TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072241-A1 4 -OXO- IH -QUINOLINE- 3 - CARBOXAMIDES AS MODULATORS OF ATP -BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-06-16 WO disclosed