SCHEMBL20109276

SCHEMBL20109276

CNCCCc1cccc(CI)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 2/20 0.43
TAAR1 Q96RJ0 2/20 0.43
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 1/20 0.43
NOS1 P29475 3/20 0.42
NOS3 P29474 2/20 0.42
NOS2 P35228 2/20 0.42
APP P05067 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
CTSK P43235 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
SLC6A4 P31645 2/20 0.36
HRH1 P35367 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL523040 0.91 KCNH2 (0.55) KCNH2MEN1KMT2ALMNATAAR1
SCHEMBL20110029 0.84 KCNH2 (0.44) KCNH2LMNATAAR1ALDH1A1ALOX15
SCHEMBL16015472 0.84 KCNH2 (0.53) KCNH2MEN1KMT2ALMNATAAR1
SCHEMBL20109296 0.79 KCNH2 (0.68) KCNH2NOS1NOS2NPSR1
SCHEMBL3630858 0.76 GRIN2D (0.44) KCNH2LMNANOS1NOS2NPSR1
SCHEMBL20109293 0.75 KCNH2 (0.55) KCNH2ALDH1A1NOS1NOS3NOS2
SCHEMBL20298968 0.75 KCNH2 (0.46) KCNH2MEN1KMT2ALMNATAAR1
SCHEMBL20109822 0.75 LMNA (0.40) MEN1KMT2ALMNATAAR1ALDH1A1
SCHEMBL20108965 0.71 MTNR1A (0.47) KCNH2NPSR1
SCHEMBL4067485 0.70 HRH3 (0.79) MEN1KMT2ALMNATAAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed