SCHEMBL20110098

SCHEMBL20110098

CCc1cc(C)nc(CCC(N)=O)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.54
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
KLF5 Q13887 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KMT2A Q03164 3/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 3/20 0.34
LMNA P02545 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
MEN1 O00255 2/20 0.33
POLB P06746 1/20 0.33
CYP1A2 P05177 1/20 0.33
IKBKB O14920 1/20 0.33
NR4A2 P43354 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16015430 0.81 HTT (0.40) HTTTP53KMT2AKDM4EALDH1A1
SCHEMBL10051192 0.74 NOS3 (0.43) HTTNOS3NOS2RAB9AKDM4E
SCHEMBL23015828 0.74 CYP1A2 (0.38) HTTTP53RAB9AKLF5SMN1; SMN2
Ammonia Solution, Strong SCHEMBL27633883 0.73 NOS3 (0.42) HTTNOS3NOS2RAB9AKDM4E
SCHEMBL2091085 0.71 HTT (1.00) HTTRAB9AKMT2AKDM4EALDH1A1
SCHEMBL1425022 0.69 HTT (0.43) HTTNOS3NOS2KMT2AKDM4E
SCHEMBL16015434 0.69 NOS3 (0.44) HTTNOS3NOS2KMT2AALDH1A1
SCHEMBL20069377 0.68 HTT (0.38) HTTKMT2AALDH1A1LMNAHSD17B10
SCHEMBL23015766 0.68 NR4A2 (0.35) HTTTP53RAB9AKLF5SMN1; SMN2
SCHEMBL5190751 0.68 ALDH1A1 (0.46) HTTSMN1; SMN2KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed