SCHEMBL20111441

SCHEMBL20111441

O=C(Nc1ncccc1O)c1cnn(-c2ccccc2)n1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.52
RAB9A P51151 9/20 0.52
ATM Q13315 1/20 0.49
HDAC1 Q13547 2/20 0.46
NTRK1 P04629 1/20 0.46
NTRK2 Q16620 1/20 0.46
NR0B1 P51843 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
USP2 O75604 1/20 0.43
HPGD P15428 1/20 0.43
XBP1 P17861 1/20 0.43
POLB P06746 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464483 0.74 HDAC1 (0.55) NPC1RAB9AHDAC1NTRK1NTRK2
SCHEMBL30648563 0.73 RAB9A (0.88) NPC1RAB9AATMNR0B1MEN1
SCHEMBL1752087 0.71 P2RX7 (0.53) NPC1RAB9AHDAC1NTRK1NTRK2
SCHEMBL1652624 0.70 NPC1 (0.61) NPC1RAB9AATMNR0B1MEN1
SCHEMBL6311452 0.69 HDAC1 (0.51) NPC1RAB9AHDAC1NTRK1NTRK2
SCHEMBL17799203 0.69 NPC1 (0.54) NPC1RAB9AATMNR0B1MEN1
SCHEMBL6399279 0.69 KDM4E (0.56) NPC1RAB9AHDAC1NTRK1NTRK2
SCHEMBL32674134 0.68 MAPT (0.59) NPC1RAB9AHDAC1NTRK1NTRK2
SCHEMBL31095864 0.68 RAB9A (0.78) NPC1RAB9AATMNR0B1MEN1
SCHEMBL18196959 0.66 RAB9A (0.69) NPC1RAB9AATMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180121597-A1 Methods to Prepare and Employ Binding Site Models for Modulation of Phosphatase Activity and Selectivity Determination ALLOSTA PHARMACEUTICALS (US) 2018-05-03 US disclosed