SCHEMBL20116196

SCHEMBL20116196

C#CCNC(=O)c1ccc(O)c(O)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.59
CA2 P00918 5/20 0.59
CA9 Q16790 5/20 0.59
CA14 Q9ULX7 5/20 0.59
CA12 O43570 4/20 0.59
HDAC6 Q9UBN7 1/20 0.55
MAOA P21397 1/20 0.54
TOP1 P11387 3/20 0.51
MAPT P10636 2/20 0.49
SNCA P37840 1/20 0.49
CA7 P43166 4/20 0.49
TERT O14746 1/20 0.49
XDH P47989 1/20 0.49
PTGS2 P35354 2/20 0.47
NAMPT P43490 1/20 0.47
JAK3 P52333 1/20 0.47
KDM4E B2RXH2 2/20 0.46
GAA P10253 2/20 0.46
POLB P06746 1/20 0.46
CA4 P22748 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28703792 0.85 CA12 (0.59) CA1CA2CA9CA14CA12
SCHEMBL11089255 0.83 HDAC6 (0.55) CA1CA2CA9CA14CA12
SCHEMBL35401735 0.82 KDM4E (0.55) CA1CA2CA9CA14CA12
SCHEMBL18083916 0.80 HDAC6 (0.60) CA1CA2CA9CA14CA12
SCHEMBL18364959 0.80 CA12 (0.65) CA1CA2CA9CA14CA12
SCHEMBL17689597 0.79 NR1H4 (0.56) CA1CA2CA9CA14CA12
SCHEMBL24379050 0.78 CA12 (0.58) CA1CA2CA9CA14CA12
SCHEMBL31366876 0.78 CA12 (0.54) CA1CA2CA9CA14CA12
SCHEMBL22231515 0.78 CA12 (0.54) CA1CA2CA9CA14CA12
SCHEMBL10029414 0.77 L3MBTL1 (0.58) CA1CA2CA9CA14CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11286231-B2 Hydrogen-bonding compounds, compositions comprising the same, and methods of preparing and using the same WAKE FOREST UNIVERSITY HEALTH SCIENCES (US) 2022-03-29 US disclosed
US-20190345096-A1 HYDROGEN-BONDING COMPOUNDS, COMPOSITIONS COMPRISING THE SAME, AND METHODS OF PREPARING AND USING THE SAME WAKE FOREST UNIVERSITY 2019-11-14 US disclosed
WO-2018081425-A1 HYDROGEN-BONDING COMPOUNDS, COMPOSITIONS COMPRISING THE SAME, AND METHODS OF PREPARING AND USING THE SAME WAKE FOREST UNIVERSITY HEALTH SCIENCES (US) 2018-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11286231-B2 Hydrogen-bonding compounds, compositions comprising the same, and methods of preparing and using the same F12, F5, F13B CA1 411/4885CA2 1334/4885CA9 245/4885
US-20190345096-A1 HYDROGEN-BONDING COMPOUNDS, COMPOSITIONS COMPRISING THE SAME, AND METHODS OF PREPARING AND USING THE SAME F12, F5, F13B CA1 443/4885CA2 1267/4885CA9 235/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.