SCHEMBL20116883

SCHEMBL20116883

CC(C)Nc1cc(-c2noc(C3CCN([S+]([O-])C4CCCCC4)CC3)n2)ccc1C=N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
CASP3 P42574 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.38
HTT P42858 2/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KIT P10721 4/20 0.37
DGAT1 O75907 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116735 0.91 SMO (0.36) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL20116682 0.86 NPC1 (0.53) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL20116688 0.84 CNR1 (0.39) SMN1; SMN2HTTGAAKITDGAT1
SCHEMBL20116798 0.82 KIT (0.42) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL20116847 0.82 NPC1 (0.42) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL20676703 0.81 LMNA (0.39) NPC1RAB9ASMN1; SMN2HTTGAA
SCHEMBL20116766 0.80 NPC1 (0.42) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL20117192 0.78 TLR9 (0.51) SMN1; SMN2HTTGAACYP3A4CYP2C9
SCHEMBL20676516 0.78 SMN1; SMN2 (0.38) NPC1RAB9ACASP3SENP7SENP6
SCHEMBL20676636 0.77 LMNA (0.46) SMN1; SMN2HTTGAAL3MBTL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed