SCHEMBL20117808

SCHEMBL20117808

CNc1cccc([C@H](CO)NC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK2 O95069 1/20 0.37
KCNA5 P22460 1/20 0.37
KCNH2 Q12809 1/20 0.37
KCNB1 Q14721 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
APP P05067 1/20 0.36
ROCK2 O75116 3/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 2/20 0.35
HIF1A Q16665 2/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRB3 P13945 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
NFKB1 P19838 1/20 0.34
DRD1 P21728 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117519 0.82 ALDH1A1 (0.49) ALDH1A1DRD3KDM4ELMNA
SCHEMBL14350620 0.80 IDO1 (0.44) MEN1KMT2AALDH1A1ADRB2ADRB1
SCHEMBL6280812 0.80 HIF1A (0.54) ALDH1A1TSHRHIF1AADRB2ADRB1
SCHEMBL4537117 0.80 IDO1 (0.44) MEN1KMT2AALDH1A1ADRB2ADRB1
SCHEMBL14262065 0.80 USP1 (0.43) ROCK2ALDH1A1LMNA
SCHEMBL24453717 0.80 USP1 (0.43) ROCK2ALDH1A1LMNA
SCHEMBL16096523 0.80 HIF1A (0.54) ALDH1A1TSHRHIF1AADRB2ADRB1
SCHEMBL6632539 0.79 CYP3A4 (0.43) KCNH2ROCK2ALDH1A1TSHRHIF1A
SCHEMBL4049006 0.79 SLC6A2 (0.43) KCNH2ALDH1A1SLC6A3GAA
Hydrochloric Acid SCHEMBL4739557 0.79 LMNA (0.56) MEN1KMT2AALDH1A1TSHRHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349990-B1 ARYL-PHENYL-SULFONAMIDE-PHENYLENE COMPOUNDS AND THEIR USE PIMCO 2664 LTD (GB) 2018-05-02 EP disclosed