SCHEMBL2011798

SCHEMBL2011798

CC(C)(C)OC(=O)N1CC[C@@H](CNC(=O)C2CCC(c3ccccc3)N(S(=O)(=O)c3ccccc3)C2)C1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
PKM P14618 1/20 0.51
TGFBR1 P36897 6/20 0.47
HTR6 P50406 3/20 0.47
BCHE P06276 2/20 0.47
TACR1 P25103 1/20 0.47
STS P08842 3/20 0.46
ACKR3 P25106 1/20 0.46
NAMPT P43490 1/20 0.44
MMP1 P03956 2/20 0.44
MMP9 P14780 2/20 0.44
MMP3 P08254 1/20 0.44
MMP7 P09237 1/20 0.44
MMP13 P45452 1/20 0.43
GPR119 Q8TDV5 1/20 0.42
MAPK8 P45983 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011799 1.00 KDM4E (0.51) KDM4EPKMTGFBR1HTR6BCHE
SCHEMBL12628193 1.00 KDM4E (0.51) KDM4EPKMTGFBR1HTR6BCHE
SCHEMBL12628523 0.96 HTR6 (0.52) KDM4EPKMTGFBR1HTR6BCHE
SCHEMBL2038075 0.96 HTR6 (0.52) KDM4EPKMTGFBR1HTR6BCHE
SCHEMBL2014458 0.96 KDM4E (0.56) KDM4EPKMTGFBR1HTR6STS
SCHEMBL12628178 0.96 KDM4E (0.56) KDM4EPKMTGFBR1HTR6STS
SCHEMBL12628525 0.86 USP30 (0.52) TGFBR1TACR1STSMMP1MMP9
SCHEMBL2012363 0.86 USP30 (0.52) TGFBR1TACR1STSMMP1MMP9
SCHEMBL12628959 0.85 STS (0.41) KDM4EPKMTGFBR1HTR6BCHE
SCHEMBL12628291 0.83 ALDH1A1 (0.44) TGFBR1TACR1STSMMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed