SCHEMBL2038075

SCHEMBL2038075

CC(C)(C)OC(=O)N1CCC[C@H](CNC(=O)C2CCC(c3ccccc3)N(S(=O)(=O)c3ccccc3)C2)C1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.52
BCHE P06276 4/20 0.52
ACKR3 P25106 1/20 0.52
KDM4E B2RXH2 1/20 0.46
PKM P14618 1/20 0.46
MMP13 P45452 2/20 0.45
MMP1 P03956 2/20 0.45
MMP9 P14780 2/20 0.45
KDM1A O60341 1/20 0.44
TGFBR1 P36897 1/20 0.44
TACR1 P25103 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KAT7 O95251 1/20 0.43
KAT8 Q9H7Z6 1/20 0.43
STS P08842 1/20 0.42
NAMPT P43490 1/20 0.42
ADAM17 P78536 1/20 0.42
MMP3 P08254 1/20 0.42
MMP7 P09237 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628523 1.00 HTR6 (0.52) HTR6BCHEACKR3KDM4EPKM
SCHEMBL2011798 0.96 KDM4E (0.51) HTR6BCHEACKR3KDM4EPKM
SCHEMBL2011799 0.96 KDM4E (0.51) HTR6BCHEACKR3KDM4EPKM
SCHEMBL12628193 0.96 KDM4E (0.51) HTR6BCHEACKR3KDM4EPKM
SCHEMBL2014458 0.91 KDM4E (0.56) HTR6KDM4EPKMTGFBR1STS
SCHEMBL12628178 0.91 KDM4E (0.56) HTR6KDM4EPKMTGFBR1STS
SCHEMBL12628959 0.83 STS (0.41) HTR6BCHEKDM4EPKMMMP13
SCHEMBL2012363 0.82 USP30 (0.52) MMP13MMP1MMP9TGFBR1TACR1
SCHEMBL12628525 0.82 USP30 (0.52) MMP13MMP1MMP9TGFBR1TACR1
SCHEMBL12628291 0.81 ALDH1A1 (0.44) MMP13MMP1MMP9TGFBR1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed