SCHEMBL20119172

SCHEMBL20119172

CN1CCc2cc(C(=O)N[SH](=O)=O)ccc2C1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.49
HDAC8 Q9BY41 3/20 0.49
WNT1 P04628 3/20 0.47
GSK3B P49841 3/20 0.47
DYRK1A Q13627 3/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
CLK2 P49760 1/20 0.45
CLK3 P49761 1/20 0.45
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
F10 P00742 1/20 0.42
DRD1 P21728 1/20 0.42
DRD5 P21918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23077104 0.84 HDAC6 (0.52) HDAC6HDAC8WNT1GSK3BDYRK1A
SCHEMBL26484688 0.83 HDAC6 (0.51) HDAC6HDAC8WNT1GSK3BDYRK1A
SCHEMBL30839551 0.79 ALDH1A1 (0.61) HDAC6HDAC8MAOAMAOBF10
SCHEMBL3313430 0.79 ALDH1A1 (0.61) HDAC6HDAC8MAOAMAOBF10
SCHEMBL12039308 0.79 MAOA (0.52) HDAC6HDAC8MAOAMAOBF10
SCHEMBL3440249 0.79 HDAC6 (0.54) HDAC6HDAC8WNT1GSK3BDYRK1A
SCHEMBL26487314 0.78 NAMPT (0.55)
SCHEMBL20119170 0.78 USP5 (0.47) HDAC6HDAC8WNT1GSK3BDYRK1A
SCHEMBL3307342 0.78 DRD1 (0.51) HDAC6HDAC8MAOAMAOBDRD1
SCHEMBL30620400 0.78 HSD17B3 (0.55) HDAC6HDAC8MAOAMAOBF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081285-A1 UREA-CONTAINING ISOXAZOLE DERIVATIVES AS FXR AGONISTS AND METHODS OF USE THEREOF ENANTA PHARMACEUTICALS, INC. (US) 2018-05-03 WO disclosed