SCHEMBL2012003

SCHEMBL2012003

C=C(c1cccc(Cl)c1)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.47
KDM4E B2RXH2 1/20 0.47
PARP1 P09874 1/20 0.47
SLC6A2 P23975 5/20 0.46
SLC6A3 Q01959 4/20 0.46
CHRNA1 P02708 2/20 0.46
CHRNG P07510 2/20 0.46
CHRNB1 P11230 2/20 0.46
CHRNB2 P17787 2/20 0.46
CHRNB4 P30926 2/20 0.46
SLC6A4 P31645 2/20 0.46
CHRNA3 P32297 2/20 0.46
CHRNA4 P43681 2/20 0.46
CHRND Q07001 2/20 0.46
ITGA5 P08648 1/20 0.46
CYP2C19 P33261 1/20 0.46
HRH1 P35367 1/20 0.46
CHRNA7 P36544 1/20 0.46
OPRK1 P41145 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8464546 0.85 KMT2A (0.39) KDM4EALDH1A1SMN1; SMN2HPGDGAA
SCHEMBL27871195 0.80 PARP1 (0.47) HTTKDM4EPARP1SLC6A2SLC6A3
SCHEMBL8081217 0.78 PARP1 (0.48) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL1361076 0.77 PARP1 (0.52) HTTKDM4EPARP1SLC6A2SLC6A3
SCHEMBL1794480 0.76 PARP1 (0.56) HTTKDM4EPARP1ALDH1A1SMN1; SMN2
SCHEMBL20148791 0.76 CES2 (0.50) PARP1SLC6A2SLC6A3CHRNB2CHRNB4
SCHEMBL18785491 0.76 LMNA (0.33) SMN1; SMN2GAAMAPT
SCHEMBL8159886 0.76 SLC6A2 (0.63) HTTKDM4EPARP1SLC6A2SLC6A3
SCHEMBL9686798 0.74 SLC6A2 (0.48) HTTKDM4EPARP1SLC6A2SLC6A3
SCHEMBL10305470 0.74 SLC6A2 (0.61) HTTPARP1SLC6A2SLC6A3CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018090006-A1 METHODS FOR DRUG DISCOVERY USING STEM CELL-DERIVED SCHWANN CELLS MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2018-05-17 WO disclosed
CN-102652159-B Stain-resistant aqueous coating composition AKZO NOBEL COATINGS INT BV 2014-08-13 CN disclosed
EP-2513237-B1 STAIN-BLOCKING AQUEOUS COATING COMPOSITION AKZO NOBEL COATINGS INT BV (NL) 2014-06-18 EP disclosed
US-8709609-B2 Stain-blocking aqueous coating composition AKZO NOVEL COATINGS INTERNATIONAL B.V. (NL) 2014-04-29 US disclosed
EP-2513237-A1 STAIN-BLOCKING AQUEOUS COATING COMPOSITION Akzo Nobel Coatings International B.V. (NL) 2012-10-24 EP disclosed
US-20120244368-A1 STAIN-BLOCKING AQUEOUS COATING COMPOSITION AKZO NOBEL COATING INTERNATIONAL B.V. (NL) 2012-09-27 US disclosed
CN-102652159-A Stain-resistant aqueous coating composition AKZO NOBEL COATINGS INT BV 2012-08-29 CN disclosed
WO-2011073164-A1 STAIN-BLOCKING AQUEOUS COATING COMPOSITION AKZO NOBEL COATINGS INTERNATIONAL B.V. (NL) 2011-06-23 WO disclosed
EP-0197274-B1 PROCESS FOR THE PREPARATION OF SUBSTITUTED STYRENES BAYER AG (DE) 1989-01-04 EP disclosed
US-4650910-A CLEAVAGE OF N-ACYL-B-PHENETHYLAMINES WITH BASE BAYER AKTIENGESELLSCHAFT (DE) 1987-03-17 US disclosed
EP-0197274-A1 Process for the preparation of substituted styrenes BAYER AG (DE) 1986-10-15 EP disclosed