SCHEMBL20120068

SCHEMBL20120068

Cc1c(CCC(=O)O)c2ccc(Br)cc2n1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.52
GPR17 Q13304 1/20 0.48
EGFR P00533 3/20 0.46
KMO O15229 1/20 0.43
PLA2G4A P47712 1/20 0.42
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
MAPT P10636 1/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
MCL1 Q07820 3/20 0.39
BCL2L1 Q07817 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PDE5A O76074 1/20 0.39
PDE9A O76083 1/20 0.39
PTGS1 P23219 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18509730 0.89 PLA2G4A (0.47) EGLN1GPR17EGFRPLA2G4AMAPT
SCHEMBL18509483 0.86 EGFR (0.49) EGFRKMOPLA2G4ATHRATHRB
SCHEMBL19872728 0.84 KDM4E (0.50) EGLN1EGFRPLA2G4ATHRATHRB
SCHEMBL19872619 0.83 MCL1 (0.55) GPR17EGFRKMOAKR1C3AKR1C2
SCHEMBL19872669 0.83 AKR1C3 (0.53) GPR17EGFRPLA2G4ATHRATHRB
SCHEMBL19872667 0.82 EGFR (0.48) EGFRPLA2G4ATHRATHRBAKR1C3
SCHEMBL25492622 0.82 EGLN1 (0.53) EGLN1GPR17KMOPLA2G4AMAPT
SCHEMBL20119990 0.81 PTGS1 (0.55) GPR17KMOAKR1C3AKR1C2KDM4E
SCHEMBL18509737 0.81 RXRA (0.54) GPR17EGFRPLA2G4ATHRATHRB
SCHEMBL21392039 0.80 FABP4 (0.45) EGFRPLA2G4ATHRATHRBAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081456-A1 HIGHLY ACTIVE SELF-SUFFICIENT NITRATION BIOCATALYSTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2018-05-03 WO disclosed