SCHEMBL20120181

SCHEMBL20120181

Cc1[nH]c2cc(-c3ccncc3)ccc2c1CCC(=O)O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 9/20 0.57
TBXAS1 P24557 1/20 0.55
EGFR P00533 1/20 0.49
APEX1 P27695 1/20 0.47
GSK3B P49841 2/20 0.45
IMPDH2 P12268 1/20 0.41
MMP2 P08253 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20120041 0.90 TBXAS1 (0.64) GPR17TBXAS1EGFRAPEX1MMP2
SCHEMBL18509728 0.88 GPR17 (0.72) GPR17EGFRAPEX1
SCHEMBL20934938 0.82 GSK3B (0.45) GPR17TBXAS1GSK3BIMPDH2MMP2
SCHEMBL18509428 0.80 EGFR (0.72) GPR17TBXAS1EGFRAPEX1
SCHEMBL18029306 0.80 IMPDH2 (0.41) GPR17TBXAS1GSK3BIMPDH2MMP2
SCHEMBL20935027 0.79 EGFR (0.56) GPR17TBXAS1EGFRAPEX1
SCHEMBL18509485 0.78 GPR17 (0.57) GPR17TBXAS1EGFRAPEX1
SCHEMBL23226279 0.78 GPR17 (0.71) GPR17EGFRAPEX1
SCHEMBL20119873 0.77 RXRA (0.45) GPR17EGFRGSK3B
SCHEMBL20935034 0.75 EGFR (0.55) GPR17TBXAS1EGFRAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081456-A1 HIGHLY ACTIVE SELF-SUFFICIENT NITRATION BIOCATALYSTS UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2018-05-03 WO disclosed