SCHEMBL20121634

SCHEMBL20121634

O=C(c1ccc(CN2CCN(C(=O)c3ccccc3)CC2)cc1)N1CCCCC1

nearest known ligand 0.81

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.76
ALDH1A1 P00352 2/20 0.76
HPGD P15428 3/20 0.70
HRH3 Q9Y5N1 3/20 0.70
LMNA P02545 2/20 0.69
SMN1; SMN2 Q16637 2/20 0.69
MEN1 O00255 2/20 0.69
KMT2A Q03164 2/20 0.69
TSHR P16473 1/20 0.69
MAPK1 P28482 1/20 0.69
L3MBTL1 Q9Y468 1/20 0.69
SIGMAR1 Q99720 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9645824 0.89 KDM4E (0.94) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL1019998 0.89 KDM4E (0.94) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL30576832 0.87 KDM4E (0.74) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL10076259 0.84 KDM4E (0.74) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL13150665 0.84 CASP1 (0.59) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL13149349 0.84 KDM4E (0.78) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL4486386 0.84 KDM4E (0.78) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL17695973 0.83 ALDH1A1 (0.68) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL19562173 0.83 KDM4E (0.68) KDM4EALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL25041158 0.82 KDM4E (0.76) KDM4EALDH1A1LMNASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963452-B2 Methods, compounds, and compositions for inhibition of ROS AUGUSTA PHARMACEUTICALS INC. (US) 2018-05-08 US disclosed