SCHEMBL2012173

SCHEMBL2012173

COc1ccncc1C(=O)N(C)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.59
HCRTR2 O43614 2/20 0.59
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ITGA4 P13612 1/20 0.40
ITGB7 P26010 1/20 0.40
PADI4 Q9UM07 3/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
HRH3 Q9Y5N1 2/20 0.37
MAPK1 P28482 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011717 1.00 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AITGA4
SCHEMBL2054013 0.84 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AITGA4
SCHEMBL2010795 0.84 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AITGA4
SCHEMBL2019129 0.83 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AITGA4
SCHEMBL2017211 0.83 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AITGA4
SCHEMBL2014804 0.83 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2013533 0.83 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AITGA4
SCHEMBL2010990 0.83 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2011939 0.83 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2053258 0.82 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9APADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed