SCHEMBL2011939

SCHEMBL2011939

COc1ccc2c(C(=O)N(C)[C@H](CCNC(=O)c3cccn3C)Cc3ccccc3)cncc2c1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.58
HCRTR2 O43614 2/20 0.58
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
TACR3 P29371 2/20 0.37
PYGL P06737 1/20 0.36
MAPT P10636 3/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 2/20 0.35
PADI4 Q9UM07 1/20 0.35
POLB P06746 1/20 0.35
CLK1 P49759 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ACHE P22303 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010990 1.00 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9ATACR3
SCHEMBL2014804 0.89 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2017401 0.84 HCRTR1 (0.70) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2016472 0.84 HCRTR1 (0.70) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2011717 0.83 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2012173 0.83 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2015123 0.82 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9AMAPT
SCHEMBL2015054 0.82 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9APYGL
SCHEMBL2015171 0.82 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AKDM4E
SCHEMBL2054419 0.82 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed