SCHEMBL20122021

SCHEMBL20122021

CC1CC2CC(C1)CC(C)(c1cc(Nc3ccc(CCC(=O)O)cc3)ccc1O)C2

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.50
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
CYP26B1 Q9NR63 2/20 0.40
CYP26A1 O43174 1/20 0.40
IDH1 O75874 11/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20122035 0.87 EPHX2 (0.47) EPHX2GSK3AGSK3BIDH1
SCHEMBL17916347 0.86 EPHX2 (0.44) EPHX2GSK3AGSK3BCYP26B1CYP26A1
SCHEMBL17911600 0.86 EPHX2 (0.57) EPHX2GSK3AGSK3BCYP26B1CYP26A1
SCHEMBL20122000 0.80 RARB (0.56) CYP26A1IDH1
SCHEMBL17911590 0.75 EPHX2 (0.52) EPHX2GSK3AGSK3B
SCHEMBL17916358 0.74 EPHX2 (0.42) EPHX2GSK3AGSK3BIDH1
SCHEMBL16517420 0.72 RARB (0.60) EPHX2
SCHEMBL20122019 0.70 EPHX2 (0.41) EPHX2GSK3AGSK3B
SCHEMBL5652618 0.69 FFAR1 (0.63)
SCHEMBL7796128 0.68 CYP26B1 (0.52) CYP26B1CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963439-B2 Specific inhibitors of cytochrome P450 26 retinoic acid hydroxylase UNIVERSITY OF WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2018-05-08 US disclosed