SCHEMBL2012216

SCHEMBL2012216

COc1cccc(C(=O)N(C)C(CCNC(=O)c2ccccn2)Cc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.47
HTR1A P08908 2/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
DRD3 P35462 1/20 0.47
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 4/20 0.43
ALOX15 P16050 1/20 0.42
KLKB1 P03952 1/20 0.41
MEN1 O00255 2/20 0.40
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011408 0.89 HCRTR1 (0.43) EPHX2HTR1AHTR2AHTR2CDRD3
SCHEMBL6919106 0.89 HCRTR1 (0.43) EPHX2HTR1AHTR2AHTR2CDRD3
SCHEMBL2017304 0.89 HCRTR1 (0.43) EPHX2HTR1AHTR2AHTR2CDRD3
SCHEMBL2016502 0.86 HCRTR1 (0.49) HTR1AHTR2AHTR2CDRD3HCRTR1
SCHEMBL13138994 0.84 KMT2A (0.55) EPHX2HCRTR1HCRTR2SMN1; SMN2ALDH1A1
SCHEMBL13138970 0.84 KMT2A (0.55) EPHX2HCRTR1HCRTR2SMN1; SMN2ALDH1A1
SCHEMBL13138974 0.84 KMT2A (0.59) EPHX2HCRTR1HCRTR2SMN1; SMN2ALDH1A1
SCHEMBL2014058 0.84 HCRTR1 (0.62) HTR1AHTR2AHTR2CDRD3HCRTR1
SCHEMBL13138991 0.84 HCRTR1 (0.60) EPHX2HTR1AHTR2ADRD3HCRTR1
SCHEMBL13138969 0.83 HCRTR1 (0.53) EPHX2HTR1AHTR2ADRD3HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed