SCHEMBL2011408

SCHEMBL2011408

COc1cccc(C(=O)NCCC(Cc2ccccc2)N(C)C(=O)c2ccnc(C)n2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.43
HCRTR2 O43614 2/20 0.43
KLKB1 P03952 1/20 0.41
CTSA P10619 1/20 0.40
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
DRD3 P35462 1/20 0.37
EPHX2 P34913 1/20 0.36
OPRM1 P35372 2/20 0.35
OPRK1 P41145 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6919106 0.91 HCRTR1 (0.43) HCRTR1HCRTR2KLKB1CTSAHTR1A
SCHEMBL2017304 0.91 HCRTR1 (0.43) HCRTR1HCRTR2KLKB1CTSAHTR1A
SCHEMBL2014681 0.89 HCRTR1 (0.43) HCRTR1HCRTR2CTSAHTR1AHTR2A
SCHEMBL2014812 0.89 HCRTR1 (0.43) HCRTR1HCRTR2CTSAHTR1AHTR2A
SCHEMBL2012216 0.89 EPHX2 (0.47) HCRTR1HCRTR2KLKB1HTR1AHTR2A
SCHEMBL2016502 0.85 HCRTR1 (0.49) HCRTR1HCRTR2KLKB1CTSAHTR1A
SCHEMBL2051291 0.84 HCRTR1 (0.43) HCRTR1HCRTR2CTSAHTR1AHTR2A
SCHEMBL2014592 0.84 HCRTR1 (0.43) HCRTR1HCRTR2CTSAHTR1AHTR2A
SCHEMBL2013880 0.83 HCRTR1 (0.46) HCRTR1HCRTR2KLKB1CTSAHTR1A
SCHEMBL2014058 0.81 HCRTR1 (0.62) HCRTR1HCRTR2KLKB1CTSAHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed