SCHEMBL2012652

SCHEMBL2012652

Fc1cccc(-c2[c]ccc(Cl)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.43
GABRD O14764 2/20 0.43
GABRA1 P14867 2/20 0.43
GABRB1 P18505 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
GABRA2 P47869 2/20 0.43
GABRB2 P47870 2/20 0.43
GABRA4 P48169 2/20 0.43
GABRE P78334 2/20 0.43
GABRA6 Q16445 2/20 0.43
GABRG1 Q8N1C3 2/20 0.43
GABRG3 Q99928 2/20 0.43
GABRQ Q9UN88 2/20 0.43
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7507597 0.86 GABRP (0.42) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1205892 0.85 TAAR1 (0.44) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL3022644 0.85 ALOX5 (0.42) TAAR1ESR2CHRNB4CHRNA3RAB9A
SCHEMBL2013527 0.83 GABRP (0.30) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1116582 0.79 GABRP (0.38) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL5106003 0.79 MAPT (0.41) MEN1KMT2AALDH1A1THRBKDM4E
SCHEMBL2431003 0.79 PTPN1 (0.39) MEN1KMT2ATAAR1ESR2NT5E
SCHEMBL1116711 0.79 CYP1A2 (0.41) MEN1KMT2AALDH1A1KDM4EMAPT
SCHEMBL7470612 0.79 TAAR1 (0.47) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2014176 0.79 ACHE (0.50) MEN1KMT2AALDH1A1THRBTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013182433-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-12-12 WO disclosed
EP-2547687-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2013-01-23 EP disclosed
EP-2513067-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2012-10-24 EP disclosed
WO-2011113820-A1 A PROCESS USING GRIGNARD REAGENTS BASF SE (DE) 2011-09-22 WO disclosed
WO-2011073145-A1 METHOD FOR PRODUCING TRIAZOLINTHIONE DERIVATIVES AND INTERMEDIATES THEREOF BASF SE (DE) 2011-06-23 WO disclosed
US-4455421-A ANTIFERTILITY, ANTIULCER AGENTS; TETRAZOLE DERIVATIVES PFIZER INC. (US) 1984-06-19 US disclosed
US-4365077-A ANTIFERTILITY, ANTIULCER PFIZER INC. (US) 1982-12-21 US disclosed
US-4157341-A 11-Desoxy-16-aryloxy-ω-tetranorprostaglandins PFIZER INC. (US) 1979-06-05 US disclosed
US-3966758-A Anti-inflammatory 1-(substituted benzyl)-2-imidazolidinones MORTON-NORWICH PRODUCTS, INC. (US) 1976-06-29 US disclosed