SCHEMBL20129615

SCHEMBL20129615

CC(C)(C)OC(=O)N=S(C)(=O)c1cccnc1Cl

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.46
ATR Q13535 1/20 0.40
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NFE2L2 Q16236 3/20 0.36
ACLY P53396 1/20 0.36
CHRM1 P11229 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
RAB9A P51151 2/20 0.34
EGFR P00533 2/20 0.34
HTT P42858 1/20 0.34
CYP2C19 P33261 1/20 0.33
METAP1 P53582 1/20 0.33
LIPE Q05469 1/20 0.33
STS P08842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21989751 0.81 PABPC1 (0.45) LMNASMN1; SMN2CHRM1RAB9AHTT
SCHEMBL20141849 0.76 EPHX2 (0.43) LMNA
SCHEMBL20129610 0.76 EPHX2 (0.43) LMNA
SCHEMBL20141065 0.76 EPHX2 (0.43) LMNA
SCHEMBL21360400 0.74 HSD11B1 (0.38) POLBSMN1; SMN2RAB9AHTT
SCHEMBL25321543 0.73 SMN1; SMN2 (0.41) POLBLMNASMN1; SMN2EGFRSTS
SCHEMBL31247697 0.73 CDK5 (0.36) LMNARAB9AHTTMETAP1
SCHEMBL24394662 0.72 CA12 (0.42) LMNARAB9ASTS
SCHEMBL3704196 0.70 COMT (0.47) POLBLMNASMN1; SMN2NFE2L2ACLY
SCHEMBL925929 0.70 NFE2L2 (0.46) LMNASMN1; SMN2NFE2L2ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2020-11-24 US disclosed
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2020-07-02 US disclosed
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
US-10414727-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2019-09-17 US disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
US-20180127370-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2018-05-10 US disclosed
US-20180127370-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2018-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof MTOR, RICTOR, RPTOR POLB 2449/4885ATR 1756/4885LMNA 3104/4885
US-10414727-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof MTOR, RICTOR, RPTOR POLB 2449/4885ATR 1756/4885LMNA 3104/4885
US-20180127370-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF MTOR, RICTOR, RPTOR POLB 2449/4885ATR 1756/4885LMNA 3104/4885
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF MTOR, RICTOR, RPTOR POLB 2449/4885ATR 1756/4885LMNA 3104/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.