SCHEMBL20133643

SCHEMBL20133643

CC1c2ccc(F)cc2C(=O)N1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
SRD5A1 P18405 3/20 0.39
PARK7 Q99497 3/20 0.39
GRIA1 P42261 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIA3 P42263 1/20 0.37
GRIA4 P48058 1/20 0.37
GPR3 P46089 1/20 0.37
P2RX7 Q99572 1/20 0.36
MC4R P32245 1/20 0.36
MC5R P33032 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
IDO1 P14902 1/20 0.35
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
ALOX5 P09917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24995868 0.80 LMNA (0.43) ACHESRD5A1GPR3CA1CA2
SCHEMBL29289807 0.79 GPR3 (0.37) GPR3
SCHEMBL22550998 0.77 MC4R (0.38) ACHEPARK7MC4RMC5R
SCHEMBL29289717 0.75 BRD4 (0.39) GPR3PGR
SCHEMBL13704120 0.73 GPR3 (0.60) GPR3
SCHEMBL22792110 0.73 GPR3 (0.60) GPR3
SCHEMBL13704044 0.73 GPR3 (0.60) GPR3
SCHEMBL30296824 0.71 PARK7 (0.35) ACHESRD5A1PARK7P2RX7CA1
SCHEMBL18863329 0.70 PIM1 (0.40) ACHEMC4RMC5RNR3C2
SCHEMBL24182508 0.70 KDM4E (0.38) GPR3P2RX7CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2020-11-24 US disclosed
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2020-07-02 US disclosed
US-10414727-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof NAVITOR PHARMACEUTICALS, INC. (US) 2019-09-17 US disclosed
US-20180127370-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. 2018-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10844013-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof MTOR, RICTOR, RPTOR ACHE 4745/4885SRD5A1 4301/4885PARK7 1844/4885
US-10414727-B2 Phenyl amino piperidine mTORC inhibitors and uses thereof MTOR, RICTOR, RPTOR ACHE 4745/4885SRD5A1 4301/4885PARK7 1844/4885
US-20180127370-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF MTOR, RICTOR, RPTOR ACHE 4745/4885SRD5A1 4301/4885PARK7 1844/4885
US-20200207716-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF MTOR, RICTOR, RPTOR ACHE 4745/4885SRD5A1 4301/4885PARK7 1844/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.