SCHEMBL2013416

SCHEMBL2013416

CN(C(=O)c1ccc2ccccc2n1)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.60
HCRTR2 O43614 2/20 0.60
NPC1 O15118 3/20 0.48
RAB9A P51151 2/20 0.48
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.39
KDM4C Q9H3R0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2015027 0.91 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2013183 0.89 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9AHTR1A
SCHEMBL2010539 0.88 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9AHPGD
SCHEMBL2016643 0.87 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2012310 0.86 HCRTR1 (0.67) HCRTR1HCRTR2NPC1RAB9AHTR1A
SCHEMBL2014058 0.84 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHTR1A
SCHEMBL13139060 0.84 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL6918071 0.83 HCRTR1 (0.66) HCRTR1HCRTR2NPC1RAB9AHTR1A
SCHEMBL2013516 0.83 HCRTR1 (0.66) HCRTR1HCRTR2NPC1RAB9AHTR1A
SCHEMBL2016503 0.83 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed