SCHEMBL2016503

SCHEMBL2016503

CN(C(=O)c1cc2ccccc2n1C)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.63
HCRTR2 O43614 2/20 0.63
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MCL1 Q07820 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011481 0.87 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AL3MBTL1
SCHEMBL13139060 0.85 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9AHDAC1
SCHEMBL2017845 0.84 HCRTR1 (0.68) HCRTR1HCRTR2NPC1RAB9AHDAC1
SCHEMBL2014120 0.84 HCRTR1 (0.68) HCRTR1HCRTR2NPC1RAB9AHDAC1
SCHEMBL2012310 0.83 HCRTR1 (0.67) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2013416 0.83 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AMEN1
SCHEMBL2011910 0.83 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9AHDAC1
SCHEMBL13139102 0.82 HCRTR1 (0.71) HCRTR1HCRTR2NPC1RAB9AHDAC1
SCHEMBL2053280 0.82 HCRTR1 (0.68) HCRTR1HCRTR2NPC1RAB9AHDAC1
SCHEMBL2049210 0.82 HCRTR1 (0.68) HCRTR1HCRTR2NPC1RAB9AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed