SCHEMBL2015027

SCHEMBL2015027

CN(C(=O)c1ccc2cnccc2n1)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.56
HCRTR2 O43614 2/20 0.56
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
PADI4 Q9UM07 3/20 0.39
CTSA P10619 2/20 0.39
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
HRH3 Q9Y5N1 2/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
GAA P10253 1/20 0.35
JAK2 O60674 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013416 0.91 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2011082 0.86 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2053258 0.86 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2013183 0.85 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2010539 0.85 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2016643 0.84 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2012310 0.82 HCRTR1 (0.67) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2019129 0.81 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2011717 0.81 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2052690 0.81 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9APADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed